huhu!
ad 1)
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serendipity:
Zufall, Bsp.: Penicillin
nach
Vorbildern aus der Natur: Pflanzen (Pilocarpin, taxol), Tiere (Tetradotoxin),
MO (Streptomycin, Tetracyclin, Penicillin)
Metabolismus:
Prodrugs
Nebenwirkungen:
Sildenafil, Disulfiram
Mimicry:
Substanzen, die den Übergangszustand simulieren (Pentostatin)
HTS: mittels
einfacher biochem. Tests bis zu 10 000 Substanzen/d untersuchbar
in silico:
durchsuchen von Datenbanken
ad 2)
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NMR, FTIR, SPR
ad 3)
jap und noch dazu moleküldynamiksimulationen
hochachtungsvoll